Chronic Conditions
Labetalol Tablets
Generic For Trandate®
starting at $24.99

Labetalol tablets are used to treat high blood pressure (hypertension) by relaxing blood vessels and slowing the heart rate. This medication works by blocking both alpha and beta receptors in the body, which helps reduce the force and rate of the heartbeat and allows blood to flow more easily. It’s often prescribed with other medications to help prevent complications like stroke, heart attack, or kidney problems caused by uncontrolled blood pressure.

  • Labetalol tablets are combined alpha- and beta-adrenergic receptor blockers
  • Should not be abruptly stopped as this may worsen heart conditions
  • Common side effects include dizziness, fatigue, and nausea
  • May be taken with or without food, but consistency is essential
HSA/FSA Eligible

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  • Labetalol Tablets Side Effects

    Labetalol tablets may cause side effects such as dizziness, fatigue, nausea, and headache, especially when starting treatment or increasing the dose. More serious side effects include slow heart rate (bradycardia), low blood pressure (hypotension), and liver function changes. Rarely, allergic reactions or heart failure symptoms may occur. Patients with asthma or other breathing problems should use labetalol cautiously, as it may worsen bronchospasm. Diabetic patients should be aware that labetalol can mask symptoms of low blood sugar. It’s important not to stop the medication suddenly, as this may lead to a rebound increase in blood pressure or heart complications.

  • Labetalol Tablets Medication Description

    Labetalol is a unique antihypertensive agent that combines selective alpha-1 adrenergic blocking and non-selective beta-adrenergic blocking properties. This dual mechanism allows it to lower blood pressure effectively by decreasing peripheral vascular resistance (via alpha blockade) and reducing heart rate and cardiac output (via beta blockade). Unlike pure beta-blockers, labetalol does not significantly reduce renal blood flow, making it a potential option in patients with kidney concerns.


    Clinically, labetalol is used to manage both chronic hypertension and hypertensive emergencies. The medication is typically started at a low dose and titrated based on blood pressure response. Because of its ability to block both alpha and beta receptors, labetalol provides a balanced approach to blood pressure control without generally causing reflex tachycardia, a common issue with pure vasodilators. It is well tolerated, but patients should be monitored for signs of bradycardia, hypotension, and liver function abnormalities during long-term use.

  • Consumer Information Use and Disclaimer

    This information should not be used to decide whether or not to take this medicine or any other medicine. Only a healthcare provider has the knowledge and training to decide which medicines are right for you. TelyRx does not endorse any medicine as safe, effective, or approved for treating any patient or health condition. This is only a limited summary of general information about the medicine’s uses from the patient education materials and is not intended to be comprehensive. This limited summary does NOT include all information about the possible uses, directions, warnings, precautions, interactions, adverse effects, or risks that may apply to this medicine. This information is not intended to provide medical advice, diagnosis or treatment and does not replace information you may receive from your healthcare provider. For a more detailed summary of information about the risks and benefits of using this medicine, please review the entire patient education information you receive with the medication.

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